| Reference: | Herrmann, J. L.; Cregge,R. J.; Richman, J. E.; Semmelhack, C. L.; Schlessinger, R. H. J. Am. Chem. Soc., 1974, 96, 3702–3703. DOI |
| Keywords: | Sulfide -> Sulfoxide • Aminal • CarboxEster enolate+Alkyl-X • CarboxCl -> CarboxAmide • N-H -> N-Alkyl • Lactam-6 • ConjAdd Enolate • CarboxAmide enolate+EnoateEster • Bischler-Napieralski • Imonium -> Amine • Amine-6 • CarboxEster -> CarboxAmide • Pummerer • |
| Reagents: | LiNiPr2 • HMPA (solvent) • TsOH • Oxalyl chloride • KH • LiNiPr2 • Acrylate • POCl3 • AlH(OtBu)3-Li+ • Perbenzoic acid, 3-chloro • NaH • Acetyl chloride • NaOMe • NaOMe • |