| Reference: | Padwa, A.; Danca, M. D.; Hardcastle, K. I.; McClure, M. S. J. Org. Chem. 2003, 68, 929-941. DOI |
| Keywords: | Sulfide -> Sulfoxide • O-SiMe2tBu -> O-H • CarboxAmide -> Thioamide • Claisen acylation, formate • CarboxEster enolate+Formate • Alkyl-OH -> Alkyl-Br • Sulfoxide-Ei -> EneLactam • Lactam -> EneLactam • CarboxAmide enolate+Alkyl-X • CarboxAmide -> Amine • Amine-5 • Aldehyde -> Enamine • Lactam-5 • Pummerer • Lactam-5 • Pictet-Spengler • |
| Reagents: | LiNiPr2 • Periodate, sodium • NaH • Periodate, sodium • Lawesson • Me3O+ X- • PPh3, CBr4 • Formate, ethyl • BH4-Na+ • Camphor sulfonic acid • |